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1

Highly Regioselective DABCO-Catalyzed Nucleophilic Aromatic Substitution (SNAr) Reaction of Methyl 2,6-Dichloronicotinate with Phenols

Yao-Jun Shi, Guy Humphrey, Peter E. Maligres, Robert A. Reamer, J. Michael Williams

Journal:

Advanced Synthesis & Catalysis

Year:

2006

Language:

english

File:

PDF, 78 KB

english, 2006

2

Development of a Second-Generation, Highly Efficient Manufacturing Route for the HIV Integrase Inhibitor Raltegravir Potassium

Humphrey, Guy R., Pye, Philip J., Zhong, Yong-Li, Angelaud, Remy, Askin, David, Belyk, Kevin M., Maligres, Peter E., Mancheno, Danny E., Miller, Ross A., Reamer, Robert A., Weissman, Steven A.

Journal:

Organic Process Research & Development

Year:

2011

Language:

english

File:

PDF, 1.22 MB

english, 2011

3

CO Cross-Coupling of Activated Aryl and Heteroaryl Halides with Aliphatic Alcohols

Peter E. Maligres, Jing Li, Shane W. Krska, John D. Schreier, Izzat T. Raheem

Journal:

Angewandte Chemie International Edition

Year:

2012

Language:

english

File:

PDF, 836 KB

english, 2012

4

High-Throughput Optimization of Ir-Catalyzed C–H Borylation: A Tutorial for Practical Applications

Preshlock, Sean M., Ghaffari, Behnaz, Maligres, Peter E., Krska, Shane W., Maleczka, Robert E., Smith, Milton R.

Journal:

Journal of the American Chemical Society

Year:

2013

Language:

english

File:

PDF, 3.00 MB

english, 2013

5

Practical, Highly Convergent, Asymmetric Synthesis of a Selective PPARγ Modulator

Maligres, Peter E., Humphrey, Guy R., Marcoux, Jean-François, Hillier, Michael C., Zhao, Dalian, Krska, Shane, Grabowski, Edward J. J.

Journal:

Organic Process Research & Development

Year:

2009

Language:

english

File:

PDF, 227 KB

english, 2009

6

Silyl Phosphorus and Nitrogen Donor Chelates for Homogeneous Ortho Borylation Catalysis

Ghaffari, Behnaz, Preshlock, Sean M., Plattner, Donald L., Staples, Richard J., Maligres, Peter E., Krska, Shane W., Maleczka, Robert E., Smith, Milton R.

Journal:

Journal of the American Chemical Society

Year:

2014

Language:

english

File:

PDF, 704 KB

english, 2014

7

A Robust Kilo-Scale Synthesis of Doravirine

Campeau, Louis-Charles, Chen, Qinghao, Gauvreau, Danny, Girardin, Mélina, Belyk, Kevin, Maligres, Peter, Zhou, Guoyue, Gu, Chaozhan, Zhang, Wei, Tan, Lushi, O’Shea, Paul D.

Journal:

Organic Process Research & Development

Year:

2016

Language:

english

File:

PDF, 347 KB

english, 2016

8

A multifunctional catalyst that stereoselectively assembles prodrugs

DiRocco, Daniel A., Ji, Yining, Sherer, Edward C., Klapars, Artis, Reibarkh, Mikhail, Dropinski, James, Mathew, Rose, Maligres, Peter, Hyde, Alan M., Limanto, John, Brunskill, Andrew, Ruck, Rebecca T.

Journal:

Year:

2017

Language:

english

File:

PDF, 777 KB

english, 2017

9

Eine neue Klasse DNA-spaltender Verbindungen: pH-abhängige DNA-Spaltung durch Propargyl- und Allenylsulfone

Prof. K. C. Nicolaou, G. Skokotas, P. Maligres, G. Zuccarello, E. J. Schweiger, K. Toshima, S. Wendeborn

Journal:

Angewandte Chemie

Year:

1989

File:

PDF, 370 KB

1989

10

Selektivität und Wirkungsmechanismus neuer DNA-spaltender Sulfone

Prof. Dr. K. C. Nicolaou, S. Wendeborn, P. Maligres, Dr. K. Isshiki, Dr. N. Zein, Dr. G. Ellestad

Journal:

Angewandte Chemie

Year:

1991

File:

PDF, 387 KB

1991

11

Endiin-Verbindungen mit säure-, base- und lichtempfindlichen Triggergruppen; chemische Simulierung der Dynemicin-A-Reaktionskaskade

Prof. K. C. Nicolaou, Dr. W.-M. Dai, S. V. Wendeborn, Dr. A. L. Smith, Dr. Y. Torisawa, P. Maligres, Dr. C.-K. Hwang

Journal:

Angewandte Chemie

Year:

1991

File:

PDF, 573 KB

1991

12

A New Class of DNA-Cleaving Molecules: pH-Dependent DNA Cleavage by Propargylic and Allenic Sulfones

Prof. K. C. Nicolaou, G. Skokotas, P. Maligres, G. Zuccarello, E. J. Schweiger, K. Toshima, S. Wendeborn

Journal:

Angewandte Chemie International Edition

Year:

1989

Language:

english

File:

PDF, 656 KB

english, 1989

13

Selectivity and Mechanism of Action of Novel DNA-Cleaving Sulfones

Prof. Dr. K. C. Nicolaou, S. Wendeborn, P. Maligres, Dr. K. Isshiki, Dr. N. Zein, Dr. G. Ellestad

Journal:

Angewandte Chemie International Edition

Year:

1991

Language:

english

File:

PDF, 638 KB

english, 1991

14

Enediyne Compounds Equipped with Acid-, Base- and Photo-Sensitive Triggering Devices. Chemical Simulation of the Dynemicin A Reaction Cascade

Prof. K. C. Nicolaou, Dr. W.-M. Dai, S. V. Wendeborn, Dr. A. L. Smith, Dr. Y. Torisawa, P. Maligres, Dr. C.-K. Hwang

Journal:

Angewandte Chemie International Edition

Year:

1991

Language:

english

File:

PDF, 565 KB

english, 1991

15

ChemInform Abstract: Nosylaziridines: Activated Aziridine Electrophiles.

P. E. MALIGRES, M. M. SEE, D. ASKIN, P. J. REIDER

Journal:

Year:

1997

File:

PDF, 30 KB

1997

16

ChemInform Abstract: Synthesis of the Orally Active Spiroindoline-Based Growth Hormone Secretagogue, MK-677.

P. E. MALIGRES, ET AL. ET AL.

Journal:

Year:

1997

File:

PDF, 28 KB

1997

17

ChemInform Abstract: Preparation of (S)-3-Carbethoxy-3-benzylpiperidine and the Growth Hormone Secretagogue L-163,540.

Peter E. Maligres, Michel M. Chartrain, Veena Upadhyay, Deborah Cohen, Robert A. Reamer, David Askin, R. P. Volante, Paul J. Reider

Journal:

Year:

1999

File:

PDF, 35 KB

1999

18

ChemInform Abstract: A Highly Catalytic Robust Palladium-Catalyzed Cyanation of Aryl Bromides.

Peter E. Maligres, Marjorie S. Waters, Fred Fleitz, David Askin

Journal:

Year:

2000

File:

PDF, 28 KB

2000

19

ChemInform Abstract: Thiol Addition to Aryl Propargyl Alcohols under Mild Conditions: An Accelerating Neighboring Group Effect.

Marjorie See Waters, Jennifer A. Cowen, J. Christopher McWilliams, Peter E. Maligres, David Askin

Journal:

Year:

2000

File:

PDF, 33 KB

2000

20

ChemInform Abstract: Stereocontrolled Preparation of a Nonpeptidal (-)-Spirobicyclic NK-1 Receptor Antagonist.

Peter E. Maligres, Marjorie M. Waters, Jaemoon Lee, Robert A. Reamer, David Askin

Journal:

Year:

2002

File:

PDF, 26 KB

2002

21

Preparation of a Clinically Investigated Ras Farnesyl Transferase Inhibitor.

Peter E. Maligres, Marjorie S. Waters, Steven A. Weissman, J. Christopher McWilliams, Stephanie Lewis, Jennifer Cowen, Robert A. Reamer, R. P. Volante, Paul J. Reider, David Askin

Journal:

Year:

2003

Language:

english

File:

PDF, 152 KB

english, 2003

22

Enantioselective Hydrogenation of α-Aryloxy α,β-Unsaturated Acids. Asymmetric Synthesis of α-Aryloxycarboxylic Acids.

Peter E. Maligres, Shane W. Krska, Guy R. Humphrey

Journal:

Year:

2004

File:

PDF, 31 KB

2004

23

Preparation of a clinically investigated ras farnesyl transferase inhibitor

Peter E. Maligres, Marjorie S. Waters, Steven A. Weissman, J. Christopher McWilliams, Stephanie Lewis, Jennifer Cowen, Robert A. Reamer, R. P. Volante, Paul J. Reider, David Askin

Journal:

Journal of Heterocyclic Chemistry

Year:

2003

Language:

english

File:

PDF, 128 KB

english, 2003

24

Diastereoselective syn-epoxidation of 2-alkyl-4-enamides to epoxyamides: Synthesis of the Merck HIV-1 protease inhibitor epoxide intermediate

P.E. Maligres, V. Upadhyay, K. Rossen, S.J. Cianciosi, R.M. Purick, K.K. Eng, R.A. Reamer, D. Askin, R.P. Volante, P.J. Reider

Journal:

Tetrahedron Letters

Year:

1995

Language:

english

File:

PDF, 236 KB

english, 1995

25

Synthesis of the orally active spiroindoline-based growth hormone secretagogue, MK-677

Peter E. Maligres, Ioannis Houpis, Kai Rossen, Audrey Molina, Jess Sager, Veena Upadhyay, Kenneth M. Wells, Robert A. Reamer, Joseph E. Lynch, David Askin, R.P. Volante, Paul J. Reider, Peter Houghton

Journal:

Year:

1997

Language:

english

File:

PDF, 706 KB

english, 1997

26

Nosylaziridines: Activated aziridine electrophiles

Peter E. Maligres, Marjorie M. See, David Askin, Paul J. Reider

Journal:

Tetrahedron Letters

Year:

1997

Language:

english

File:

PDF, 271 KB

english, 1997

27

A highly catalytic robust palladium catalyzed cyanation of aryl bromides

Peter E. Maligres, Marjorie S. Waters, Fred Fleitz, David Askin

Journal:

Tetrahedron Letters

Year:

1999

Language:

english

File:

PDF, 240 KB

english, 1999

28

Thiol addition to aryl propargyl alcohols under mild conditions: an accelerating neighboring group effect

Marjorie See Waters, Jennifer A Cowen, J.Christopher McWilliams, Peter E Maligres, David Askin

Journal:

Tetrahedron Letters

Year:

2000

Language:

english

File:

PDF, 167 KB

english, 2000

29

A new designed tumor selective daunomycin derivative

P.E. Maligres, K.C. Nicolaou, W. Wrasidlo

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1993

Language:

english

File:

PDF, 331 KB

english, 1993

30

Cyclic imidate salts in acyclic stereochemistry: Diastereoselective syn-epoxidation of 2-alkyl-4-enamides to epoxyamides

P.E. Maligres, S.A. Weissman, V. Upadhyay, S.J. Cianciosi, R.A. Reamer, R.M. Purick, J. Sager, K. Rossen, K.K. Eng, D. Askin, R.P. Volante, P.J. Reider

Journal:

Year:

1996

Language:

english

File:

PDF, 821 KB

english, 1996

31

Development of a Kilogram-Scale Asymmetric Synthesis of a Potent DP Receptor Antagonist

Tudge, Matthew, Savarin, Cecile G., DiFelice, Katherine, Maligres, Peter, Humphrey, Guy, Reamer, Bob, Tellers, David M., Hughes, Dave

Journal:

Organic Process Research & Development

Year:

2010

Language:

english

File:

PDF, 909 KB

english, 2010

32

ChemInform Abstract: Cyclic Imidate Salts in Acyclic Stereochemistry: Diastereoselective syn-Epoxidation of 2-Alkyl-4-enamides to Epoxyamides.

P. E. MALIGRES, S. A. WEISSMAN, V. UPADHYAY, S. J. CIANCIOSI, R. A. REAMER, R. M. PURICK, J. SAGER, K. ROSSEN, K. K. ENG, D. ASKIN, R. P. VOLANTE, P. J. REIDER

Journal:

Year:

1996

File:

PDF, 30 KB

1996

33

Porcine liver esterase-catalyzed enantioselective hydrolysis of a prochiral diester into its optically pure (S)-ester acid, a precursor to a growth hormone secretagogue

Michel Chartrain, Peter Maligres, Deborah Cohen, Veena Upadhyay, Victor Pecore, David Askin, Randolph Greasham

Journal:

Journal of Bioscience and Bioengineering

Year:

1999

Language:

english

File:

PDF, 412 KB

english, 1999

34

A Soluble Copper(I) Source and Stable Salts of Volatile Ligands for Copper-Catalyzed C–X Couplings

Maligres, Peter E., Krska, Shane W., Dormer, Peter G.

Journal:

Journal of Organic Chemistry

Year:

2012

Language:

english

File:

PDF, 414 KB

english, 2012

35

CO Cross-Coupling of Activated Aryl and Heteroaryl Halides with Aliphatic Alcohols

Peter E. Maligres, Jing Li, Shane W. Krska, John D. Schreier, Izzat T. Raheem

Journal:

Angewandte Chemie

Year:

2012

Language:

english

File:

PDF, 825 KB

english, 2012

36

ChemInform Abstract: A Soluble Copper(I) Source and Stable Salts of Volatile Ligands for Copper-Catalyzed C-X Couplings.

Maligres, Peter E., Krska, Shane W., Dormer, Peter G.

Journal:

Year:

2013

File:

PDF, 43 KB

2013

37

DNA-cleavage and antitumor activity of designed molecules with conjugated phosphine oxide-allene-ene-yne functionalities

Nicolaou, K. C., Maligres, P., Shin, J., De Leon, E., Rideout, Darryl

Journal:

Journal of the American Chemical Society

Year:

1990

Language:

english

File:

PDF, 264 KB

english, 1990

38

Stereocontrolled Preparation of a Nonpeptidal (−)-Spirobicyclic NK-1 Receptor Antagonist

Maligres, Peter E., Waters, Marjorie M., Lee, Jaemoon, Reamer, Robert A., Askin, David, Ashwood, Michael S., Cameron, Mark

Journal:

Journal of Organic Chemistry

Year:

2002

Language:

english

File:

PDF, 149 KB

english, 2002

39

Preparation of ( S )-3-Carbethoxy-3-benzylpiperidine and the Growth Hormone Secretagogue L-163,540

Maligres, Peter E., Chartrain, Michel M., Upadhyay, Veena, Cohen, Deborah, Reamer, Robert A., Askin, David, Volante, R. P., Reider, Paul J.

Journal:

Journal of Organic Chemistry

Year:

1998

Language:

english

File:

PDF, 63 KB

english, 1998

40

Enantioselective Hydrogenation of α-Aryloxy α,β-Unsaturated Acids. Asymmetric Synthesis of α-Aryloxycarboxylic Acids

Maligres, Peter E., Krska, Shane W., Humphrey, Guy R.

Journal:

Organic Letters

Year:

2004

Language:

english

File:

PDF, 52 KB

english, 2004

41

A Traceless Directing Group for CH Borylation

Preshlock, Sean M., Plattner, Donald L., Maligres, Peter E., Krska, Shane W., Maleczka, Robert E., Smith, Milton R.

Journal:

Angewandte Chemie International Edition

Year:

2013

Language:

english

File:

PDF, 408 KB

english, 2013

42

Enantioselective Synthesis of an HCV NS5a Antagonist

Mangion, Ian K., Chen, Cheng-yi, Li, Hongmei, Maligres, Peter, Chen, Yonggang, Christensen, Melodie, Cohen, Ryan, Jeon, Ingyu, Klapars, Artis, Krska, Shane, Nguyen, Hoa, Reamer, Robert A., Sherry, Ben

Journal:

Organic Letters

Year:

2014

Language:

english

File:

PDF, 536 KB

english, 2014

43

Molecular design and chemical synthesis of potent enediynes. 1. Dynemicin model systems equipped with N-tethered triggering devices

Nicolaou, K. C., Maligres, P., Suzuki, T., Wendeborn, S. V., Dai, W. M., Chadha, R. K.

Journal:

Journal of the American Chemical Society

Year:

1992

Language:

english

File:

PDF, 2.50 MB

english, 1992

44

Synthesis of a β-Amino Acid Pharmacophore via a β-Lactam Intermediate

Angelaud, Rémy, Zhong, Yong-Li, Maligres, Peter, Lee, Jaemoon, Askin, David

Journal:

Journal of Organic Chemistry

Year:

2005

Language:

english

File:

PDF, 107 KB

english, 2005

45

Asymmetric Synthesis of Cyclic Indole Aminals via 1,3-Stereoinduction

Li, Hongmei, Chen, Cheng-yi, Nguyen, Hoa, Cohen, Ryan, Maligres, Peter E., Yasuda, Nobuyoshi, Mangion, Ian, Zavialov, Ilia, Reibarkh, Mikhail, Chung, John Y. L.

Journal:

Journal of Organic Chemistry

Year:

2014

Language:

english

File:

PDF, 929 KB

english, 2014

46

Synthesis of Prostaglandin D 2 Receptor Antagonist

Tudge, M., Savarin, C., DiFelice, K., Maligres, P., Humphrey, G., Reamer, B., Tellers, D., Hughes, D.

Journal:

Year:

2010

Language:

english

File:

PDF, 99 KB

english, 2010

47

Synthesis of a Selective PPARγ Modulator

P. Maligres, G. Humphrey, J. Marcoux, M. Hillier, D. Zhao, S. Krska, E. Grabowski

Year:

2009

Language:

english

File:

PDF, 73 KB

english, 2009

48

Enantioselective Synthesis of α-Methyl-β-Cyclopropyldihydrocinnamates

Christensen, Melodie, Nolting, Andrew, Shevlin, Michael, Weisel, Mark, Maligres, Peter E., Lee, Joshua, Orr, Robert K, Plummer, Christopher W., Tudge, Matthew Thomas, Campeau, Louis-Charles, Ruck, Reb

Journal:

Journal of Organic Chemistry

Year:

2016

Language:

english

File:

PDF, 670 KB

english, 2016

49

An approach to heterodiarylmethanes via sp2-sp3 Suzuki−Miyaura cross-coupling

Stewart, Gavin W., Maligres, Peter E., Baxter, Carl A., Junker, Ellyn M., Krska, Shane W., Scott, Jeremy P.

Journal:

Year:

2016

Language:

english

File:

PDF, 920 KB

english, 2016

50

A Synthesis of a Spirocyclic Macrocyclic Protease Inhibitor for the Treatment of Hepatitis C

Chung, Cheol K., Cleator, Ed, Dumas, Aaron M., Hicks, Jacqueline D., Humphrey, Guy R., Maligres, Peter E., Nolting, Andrew F., Rivera, Nelo, Ruck, Rebecca T., Shevlin, Michael

Journal:

Organic Letters

Year:

2016

Language:

english

File:

PDF, 529 KB

english, 2016